Danazol Binding to Rat Androgen, Glucocorticoid, Progesterone, and Estrogen Receptors: Correlation With Biologic Activity
This study investigated the binding affinities of danazol to rat androgen, glucocorticoid, progesterone, and estrogen receptors and correlated these findings with the drug's known biological activity.
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Cited by (50)
- Danazol alters mitochondria metabolism of fibrocystic breast Mcf10A cells 2017
- Efectos del danazol y hemisuccinato de danazol sobre la presión de perfusión y resistencia vascular 2010
- Progestins for the Treatment of Endometriosis: An Update: 2010
- Progestins for the Treatment of Endometriosis: An Update 2010
- Local application of danazol-loaded hyaluronic acid hydrogel to endometriosis in a rat model 2006
- Treatment of Endometrial Hyperplasia with a Danazol-Releasing Intrauterine Device: A Prospective Study 2004
- A Benefit-Risk Assessment of Medical Treatment for Uterine Leiomyomas 2002
- Danazol mimics antigestagen action in first trimester termination of pregnancy 2001
- Altered uterine artery blood flow impedance after danazol therapy: possible mode of action in dysfunctional uterine bleeding 1999
- Hormone replacement therapy following hysterectomy for endometriosis 1998
- Danazol administration after gonadotrophin-releasing hormone analogue reduces rebound of uterine myomas [published erratum appears in Hum Reprod 1998 Mar;13(3):780] 1997
- Expression of Aromatase Cytochrome P450 Protein and Messenger Ribonucleic Acid in Human Endometriotic and Adenomyotic Tissues but not in Normal Endometrium1 1997
- Danazol concentrations in ovary, uterus, and serum and their effect on the hypothalamic-pituitary-ovarian axis during vaginal administration of a danazol suppository 1995
- Pain recurrence: A quality of life issue in endometriosis 1995
- Leukocyte Subpopulation Changes in Rats With Autotransplanted Endometrium and the Effect of Danazol 1995
- In utero virilization by danazol: Effects on adrenal steroidogenesis 1995
- [<sup>3</sup>H]Dexamethasone Binding Activity in Liver Microsomes is Modulated Differently by 17 α‐Alkylated Androgens and Testosterone<i>in vivo</i> 1995
- Stanozolol and danazol, unlike natural androgens, interact with the low affinity glucocorticoid-binding sites from male rat liver microsomes. 1994
- Goserelin (Zoladex) versus danazol for endometriosis: the North American experience 1994
- Induction of true precocious puberty by neonatal treatment with danazol in female rats 1993
- The effects of fetal exposure to danazol 1992
- Ambiguedad sexual por exposición a DANAZOL 1992
- Estrogen binding capacity in cytosol fraction of human uterine cervix: effect of estrogen and anti-estrogens 1992
- Thermoregulatory and endocrine effects of a low dose of danazol in postmenopausal women: Interaction with the effect of naloxone 1991
- Elimination of ovulation and menstrual cyclicity (with danazol) improves dysphoric premenstrual syndromes 1991
- The use of danazol as a treatment of endometriosis 1991
- Effects of an androgenic derivative on pre-established mammary tumours chemically induced in the rat 1991
- Elimination of ovulation and menstrual cyclicity (with danazol) improves dysphoric premenstrual syndromes. 1991
- Medical treatment of mild endometriosis associated with infertility 1991
- Comparison of the pharmacology of nafarelin and danazol 1990
- Endometriosis 1990 1990
- Cyclic Pelvic Pain 1990
- Danazol concentrations in human ovarian follicular fluid and their relationship to simultaneous serum concentrations 1988
- New Therapy for Endometriosis 1988
- Effect of progestins, androgens, estrogens and antiestrogens on3H-thymidine uptake by human endometrial and endosalpinx cells in vitro 1987
- Immunosuppressive effects of danazol in vitro 1987
- Pelvic Endometriosis 1987
- Growth inhibition by danazol in a human endometrial cancer cell line with estrogen-independent progesterone receptors 1987
- Cytoplasmic and nuclear estrogen binding capacity in the rat uterus during treatment with danazol and testosterone 1986
- Inhibition of gonadotropin-releasing hormone receptors in rat anterior pituitary monolayer cell cultures by danazol 1986
- Gestrinone (R2323) Binding to Steroid Receptors in Human Uterine Endometrial Cytosol 1986
- Danazol binds to progesterone receptors and inhibits the growth of human endometrial cancer cells in vitro 1986
- Ultrastructural changes in endometriotic tissue during danazol treatment 1985
- Danazol plus testosterone enanthate in male langur monkey 1985
- Gynecologic Problems of Adolescence 1985
- Serum estradiol and danazol. I. Endometriosis response, side effects, administration interval, concurrent spironolactone and dexamethasone 1985
- Danazol in the treatment of endometriosis: analysis of 100 cases with a 4-year follow-up 1985
- Short‐term effects of danazol on endometrial histology 1984
- Cytosol estrogen and progestin receptor concentrations and 17β‐hydroxysteroid dehydrogenase activities in the endometrium and endometriotic tissue 1984
- Regression of endometriosis following shorter treatment with, or lower dose of danazol: Comparison of pre‐ and post‐treatment laparoscopic findings in the Scandinavian multi‐center study 1984
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