Schiele F

ORCID: 0000-0002-1922-2696 · 1 paper in corpus
lab-animal 2016
British journal of pharmacology ·doi:10.1111/bph.13342

BACKGROUND AND PURPOSE: Drug-target residence time is an important, yet often overlooked, parameter in drug discovery. Multiple studies have proposed an increased residence time to be beneficial for improved drug efficacy and/or longer dura…