CULLINAN George J.

The present invention provides novel, reduced benzothiophenes of formula IwhereinR is -H, -OH, -O(C1-C4 alkyl), -O-CO-(C1-C6 alkyl), -O-CO-Ar in which Ar is optionally substituted phenyl, or -O-SO2-(C4-C6 alkyl);Ris -H, -OH, -O(C1-C4 alkyl)…

The present invention provides method of treating endometriosis using novel benzothiophene compounds of formula IwhereinR is -H, -OH, -O(C1-C4 alkyl), -O-CO-(C1-C6 alkyl), -O-CO-Ar in which Ar is optionally substituted phenyl, or -O-SO2-(…

The present invention provides a compound of formula I (I) wherein R1 is hydrogen, a hydroxy protecting group, or methyl; R2 and R3 are independently C1-C6 alkyl, or R2 and R3, together with the nitrogen to which they are attached, form…

A method of inhibiting endometriosis comprising administering to a human in need of treatment an effective amount of a compound having the formula (I) Wherein R1 and R3 are independently hydrogen, -CH3, wherein Ar is optionally su…

The present invention provides derivatives of 2-phenylmethyl-3-[4-(2-aminoethoxy)phenyl]-benzo[b]thiophene. The present invention further provides pharmaceutical compositions containing these derivatives and the use of such compounds alone,…

The present invention provides a compound of formula I I wherein R1 is -H, -OH, -O(C1-C4 alkyl), -OCOC6H5, -OCO(C1-C6 alkyl), or -OSO2 (C4-C6 alkyl); R2 is -H, -OH, -O(C1-C4 alkyl), -OCOC6H5, -OCO(C1-C6 alkyl) or -OSO2 (C4-C6 alkyl); n …