The present invention provides novel benzofuran compound, pharmaceutical formulations and processes for preparation thereof, and methods of using such compounds for alleviating the symtoms of post-menopausal syndrome, and inhibiting endomet…
The present invention provides novel benzothiophene compounds, pharmaceutical formulations, and processes for preparation thereof, and methods of using such compounds for alleviating the symptoms of post-menopausal syndrome and inhibiting e…
The present invention provides a compound of formula I wherein R1 is H, OH, halo, OCO(C1-C6 alkyl), OCO(aryl), OSO2(C4-C6 alkyl), OCOO(C1-C6 alkyl), OCOO(aryl), OCONH(C1-C6 alkyl), or OCON(C1-C6 alkyl)2; R2 is aryl, C1-C6 alkyl, C3-C6 cyc…
The present invention provides benzothiophene compounds with nitrogen-containing non-basic side chains. The present invention also provides pharmaceutical compositions containing said compounds, optionally containing estrogen or progestin, …
The present invention provides compounds with nitrogen-containing non-basic side chains of formula II. The present invention also provides pharmaceutical compositions containing compounds of formula II, optionally containing estrogen or pro…
The present invention provides compounds with nitrogen-containing non-basic side chains. The present invention also provides pharmaceutical compositions containing said compounds, optionally containing estrogen or progestin, and the use of …
The present invention provides certain novel naphthyl and dihydro compounds which are useful for alleviating the symptoms of post-menopausal syndrome, including osteoporosis, hyperlipidemia, and estrogen-dependent cancer, and inhibiting ute…
The present invention provides a compound of formula I wherein R is -H, -OH, -O(C -C alkyl), -OCOC H , -OCO(C -C alkyl), or -OSO (C -C alkyl); R² is -H, -OH, -O(C -C alkyl), -OCOC H , -OCO(C -C alkyl) or -OSO (C -C alkyl); n is 2 or 3; and…
The present invention provides a compound of formula I wherein R1 is H, OH, halo, OCO(C1-C6 alkyl), OCO(aryl), OSO2(C4-C6 alkyl), OCOO(C1-C6 alkyl), OCOO(aryl), OCONH(C1-C6 alkyl), or OCON(C1-C6 alkyl)2; R2 is aryl, C1-C6 alkyl, C3-C6 cyc…